TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 730nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 730nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 940nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 940nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.78E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: 1.78E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataKi: >2.23E+3nMAssay Description:Inhibition of P-glycoprotein in human drug-resistant K562/ADR cells assessed as reduction in P-gp mediated rhodamine 123 efflux by spectrofluorometryMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.690nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.910nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair